SCHEMBL2421099

SCHEMBL2421099

O=[N+]([O-])c1ccc(CCP(=O)(O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.61
AKR1C3 P42330 1/20 0.57
KCNJ1 P48048 4/20 0.54
KCNH2 Q12809 3/20 0.54
HRH3 Q9Y5N1 1/20 0.51
LOXL2 Q9Y4K0 1/20 0.50
CA1 P00915 2/20 0.49
CYP2C19 P33261 2/20 0.49
CA12 O43570 1/20 0.49
MMP2 P08253 1/20 0.49
MMP9 P14780 1/20 0.49
MMP8 P22894 1/20 0.49
MMP14 P50281 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CA2 P00918 1/20 0.49
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
POLB P06746 1/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28588668 0.83 TSHR (0.54) TSHRAKR1C3KCNJ1KCNH2HRH3
SCHEMBL28506967 0.82 GRIN2D (0.55) TSHRALDH1A1
SCHEMBL7610991 0.81 TSHR (0.56) TSHRAKR1C3KCNJ1KCNH2HRH3
SCHEMBL916699 0.81 AKR1C3 (0.61) TSHRAKR1C3LOXL2CA1CYP2C19
SCHEMBL7914116 0.80 CFTR (0.53) TSHRAKR1C3KCNJ1KCNH2HRH3
SCHEMBL3292782 0.80 TSHR (0.75) TSHRKCNJ1KCNH2HRH3LOXL2
SCHEMBL8094543 0.78 POLB (0.68) TSHRKCNJ1KCNH2HRH3LOXL2
SCHEMBL735219 0.77 AKR1C3 (0.61) TSHRAKR1C3KCNJ1KCNH2HRH3
Phosphoric Acid SCHEMBL28639141 0.77 CA1 (0.65) TSHRAKR1C3CA1CA12MMP2
SCHEMBL7914124 0.77 SMN1; SMN2 (0.52) TSHRAKR1C3CYP2C19ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110224096-A1 FLUORESCENT PHOSPHONIC ESTER LIBRARY TECHNISCHE UNIVERSITAT GRAZ (AT) 2011-09-15 US disclosed
WO-2010010017-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-01-28 WO disclosed
US-20080108508-A1 Fluorescent Phosphonic Ester Library TECHNISCHE UNIVERSITÄT GRAZ (AT) 2008-05-08 US disclosed
EP-1771735-A1 FLUORESCENT PHOSPHONIC ESTER LIBRARY Technische Universität Graz (AT) 2007-04-11 EP disclosed
WO-2006010403-A1 FLUORESCENT PHOSPHONIC ESTER LIBRARY TECHNISCHE UNIVERSITÄT GRAZ (AT) 2006-02-02 WO disclosed