SCHEMBL2421340

SCHEMBL2421340

CCC[C@H](N)C(=O)NC1CC[C@H]2CN(S(=O)(=O)c3ccc(C(F)(F)F)cc3)CC12

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 18/20 0.81
GAA P10253 1/20 0.45
KCNH2 Q12809 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16498680 1.00 CACNA1B (0.81) CACNA1BGAAKCNH2
SCHEMBL66748 1.00 CACNA1B (0.81) CACNA1BGAAKCNH2
SCHEMBL65962 1.00 CACNA1B (0.81) CACNA1BGAAKCNH2
SCHEMBL66758 0.91 CACNA1B (0.83) CACNA1BGAAKCNH2
SCHEMBL66453 0.90 CACNA1B (1.00) CACNA1BGAAKCNH2
SCHEMBL2419596 0.90 CACNA1B (1.00) CACNA1BGAAKCNH2
SCHEMBL16498044 0.89 CACNA1B (0.85) CACNA1BGAAKCNH2
SCHEMBL2421678 0.89 CACNA1B (0.85) CACNA1BGAAKCNH2
SCHEMBL65323 0.89 CACNA1B (0.85) CACNA1BGAAKCNH2
SCHEMBL66593 0.89 CACNA1B (0.85) CACNA1BGAAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367790-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS Abbott Laboratories (US) 2011-09-28 EP claimed
WO-2011149995-A1 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA [C]PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed