SCHEMBL24248259

SCHEMBL24248259

NC(=O)c1nc(-c2ccccc2)cnc1N

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ATR Q13535 18/20 0.67
PRKDC P78527 5/20 0.67
IKBKB O14920 1/20 0.64
ATM Q13315 2/20 0.61
MAP2K3 P46734 1/20 0.61
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3462610 0.97 ATR (0.63) ATRPRKDCIKBKBATMMAP2K3
SCHEMBL3460420 0.90 ASIC3 (0.63) ATRPRKDCIKBKBATM
SCHEMBL318797 0.88 ATR (0.68) ATRPRKDCIKBKBATMCYP3A4
SCHEMBL20433206 0.86 ATR (0.67) ATRIKBKBCYP3A4
Hydrochloric Acid SCHEMBL28324236 0.85 IKBKB (0.58) ATRPRKDCIKBKBATMMAP2K3
SCHEMBL14525246 0.85 ATR (0.65) ATRPRKDCATMCYP3A4
SCHEMBL3460235 0.85 ATR (0.70) ATRPRKDC
SCHEMBL3460497 0.84 ATR (0.71) ATRPRKDCATM
SCHEMBL18895999 0.84 ATR (0.64) ATRPRKDCIKBKBATM
SCHEMBL5684569 0.84 ATR (0.63) ATRPRKDCATMCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3354650-B1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2022-02-16 EP disclosed