SCHEMBL24253938

SCHEMBL24253938

O=C1CCCC2(CCN(c3cc(-n4cc(C(F)(F)F)cn4)ncn3)CC2)N1c1ccc(F)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC34A1 Q06495 4/20 0.34
MOGAT2 Q3SYC2 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
KCNH2 Q12809 1/20 0.31
LTC4S Q16873 1/20 0.31
DPP4 P27487 2/20 0.31
MLYCD O95822 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30424472 1.00 SLC34A1 (0.34) SLC34A1MOGAT2HCRTR1HCRTR2KCNH2
SCHEMBL24253834 0.90 HCRTR1 (0.33) HCRTR1HCRTR2KCNH2LTC4SDPP4
SCHEMBL24253540 0.90 HCRTR1 (0.34) HCRTR1HCRTR2KCNH2LTC4SDPP4
SCHEMBL24253937 0.89 CYP1A2 (0.35) HCRTR1HCRTR2KCNH2LTC4SDPP4
SCHEMBL24253900 0.88 PDE10A (0.32) MOGAT2HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL24253731 0.88 MOGAT2 (0.33) MOGAT2HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL24253628 0.87 HCRTR1 (0.31) HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL30423610 0.87 HCRTR1 (0.31) HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL24253544 0.86 HCRTR1 (0.31) HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL30423848 0.86 HCRTR1 (0.31) HCRTR1HCRTR2KCNH2LTC4S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2022-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof REN, NR3C2, PKD1 SLC34A1 112/4885MOGAT2 4470/4885HCRTR1 2245/4885
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF REN, NR3C2, PKD1 SLC34A1 112/4885MOGAT2 4470/4885HCRTR1 2245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.