SCHEMBL24254413

SCHEMBL24254413

N#Cc1ccc(C2OCCO2)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.44
ABCB1 P08183 3/20 0.39
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
CHRND Q07001 1/20 0.39
MEN1 O00255 1/20 0.37
TTR P02766 1/20 0.37
ALB P02768 1/20 0.37
KMT2A Q03164 1/20 0.37
EGLN2 Q96KS0 1/20 0.35
ELANE P08246 4/20 0.34
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25383534 0.79 ABCB1 (0.39) ABCB1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL16441689 0.77 CYP11B2 (0.50) CYP11B2CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL30976421 0.77 CYP11B2 (0.50) CYP11B2CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL30826553 0.74 PDE4B (0.44) MEN1KMT2AKDM4E
SCHEMBL21241613 0.74 PDE4B (0.44) MEN1KMT2AKDM4E
SCHEMBL17202430 0.74 CYP11B2 (0.48) CYP11B2CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL122002 0.73 CYP11B2 (0.43) CYP11B2CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL31725635 0.73 KDM1A (0.34) CHRNB2CHRNB4CHRNA3CHRNA4MEN1
SCHEMBL31725748 0.73 MAP3K14 (0.39) CHRNB2CHRNA4HTT
SCHEMBL12656462 0.73 KDM1A (0.34) CHRNB2CHRNB4CHRNA3CHRNA4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022035763-A1 BORON CONTAINING COMPOUNDS AND THEIR USES 5METIS, INC. (US) 2022-02-17 WO disclosed
WO-2022035763-A1 BORON CONTAINING COMPOUNDS AND THEIR USES 5METIS, INC. (US) 2022-02-17 WO disclosed