SCHEMBL24254493

SCHEMBL24254493

Cc1ccc(S(=O)(=O)Nc2ccc(-n3ccnc3)cc2)cc1C(=O)NCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.50
CYP2D6 P10635 2/20 0.50
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50
APH1A Q96BI3 1/20 0.50
PSENEN Q9NZ42 1/20 0.50
MAPK1 P28482 1/20 0.49
MAPT P10636 4/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 3/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24254525 0.81 CYP3A4 (0.50) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL26188253 0.79 CYP3A4 (0.48) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL24254492 0.73 NPC1 (0.61) MAPTALDH1A1LMNAMEN1KMT2A
SCHEMBL24254524 0.72 CYP3A4 (0.61) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL7129269 0.69 CYP3A4 (0.59) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL9262065 0.66 PSEN1 (0.69) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL21246574 0.66 ALDH1A1 (0.70) ALDH1A1MEN1KMT2AHTTNAMPT
SCHEMBL4880963 0.66 CYP3A4 (0.64) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL26188514 0.66 CYP3A4 (0.45) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL7129864 0.65 CYP3A4 (0.66) CYP3A4CYP2D6PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022035804-A1 SUBSTITUTED 3-AMINO-4-METHYLBENZENESULFONAMIDES AS SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-02-17 WO disclosed