SCHEMBL24255521

SCHEMBL24255521

Cc1cc2cn(C)nc2cc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 2/20 0.43
NSD2 O96028 1/20 0.43
STIM1 Q13586 2/20 0.34
ORAI1 Q96D31 2/20 0.34
NOTUM Q6P988 2/20 0.33
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
MAOA P21397 2/20 0.30
MAOB P27338 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19531676 0.93 ALDH1A1 (0.43) ALDH1A1MAPTKDM4ENSD2STIM1
SCHEMBL24163748 0.84 KDM4E (0.42) ALDH1A1MAPTKDM4ENSD2STIM1
SCHEMBL31714344 0.81 MAPT (0.42) ALDH1A1MAPTKDM4ENSD2
SCHEMBL15730121 0.81 KDM4E (0.52) ALDH1A1MAPTKDM4ENSD2STIM1
SCHEMBL29318295 0.79 MAPT (0.41) ALDH1A1MAPTKDM4ENSD2MAOA
SCHEMBL29318392 0.79 MAPT (0.41) ALDH1A1MAPTKDM4ENSD2MAOA
SCHEMBL29303280 0.78 KDM4E (0.40) ALDH1A1MAPTKDM4ENSD2NOTUM
SCHEMBL24255256 0.77 MAPT (0.42) ALDH1A1MAPTKDM4ENSD2STIM1
SCHEMBL24930081 0.77 KDM4E (0.42) ALDH1A1MAPTKDM4ENSD2STIM1
SCHEMBL26482518 0.77 MAPT (0.42) ALDH1A1MAPTKDM4ENSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022036177-A1 ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2022-02-17 WO disclosed