SCHEMBL24256714

SCHEMBL24256714

CCCc1ccc2c(N)c(C(=O)NCCc3ccc(OCCc4ccc5c(N)c(C(=O)NCCc6ccc(N7CCNCC7)cc6)sc5n4)c(OC)c3)sc2n1

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
USP28 Q96RU2 18/20 0.69
USP25 Q9UHP3 17/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24256673 0.84 MTOR (0.59) USP28USP25
SCHEMBL22957256 0.83 USP28 (0.85) USP28USP25
SCHEMBL22957383 0.82 USP28 (1.00) USP28USP25
SCHEMBL22957479 0.81 USP28 (1.00) USP28USP25
SCHEMBL22957254 0.81 USP25 (1.00) USP28USP25
SCHEMBL22957376 0.79 USP28 (1.00) USP28USP25
SCHEMBL22957316 0.79 USP25 (1.00) USP28USP25
SCHEMBL22957278 0.78 USP25 (1.00) USP28USP25
SCHEMBL22957398 0.78 USP28 (1.00) USP28USP25
SCHEMBL22957508 0.77 USP25 (1.00) USP28USP25

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022035806-A1 FUSED TRICYCLIC PYRIMIDINE-THIENO-PYRIDINE SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-02-17 WO disclosed