SCHEMBL24257707

SCHEMBL24257707

N#Cc1ncc(-c2cccc(Cl)c2)c(C(F)F)c1OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.40
SQOR Q9Y6N5 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GRM5 P41594 2/20 0.37
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
PTGER1 P34995 4/20 0.36
CYP2C9 P11712 2/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
CYP3A4 P08684 1/20 0.36
PGGT1B P53609 1/20 0.36
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30452556 1.00 CNR1 (0.40) CNR1SQORGABRG2GABRB3GABRA5
SCHEMBL24257771 0.84 GRM5 (0.42) CNR1SQORGABRG2GABRB3GABRA5
SCHEMBL30452737 0.84 GRM5 (0.42) CNR1SQORGABRG2GABRB3GABRA5
SCHEMBL30453193 0.80 GRM5 (0.42) CNR1SQORGABRG2GABRB3GABRA5
SCHEMBL24257765 0.80 GRM5 (0.42) CNR1SQORGABRG2GABRB3GABRA5
SCHEMBL24257841 0.80 LRRK2 (0.43) ADORA2AADORA1GRM5KDM4EALDH1A1
SCHEMBL30453863 0.80 LRRK2 (0.43) ADORA2AADORA1GRM5KDM4EALDH1A1
SCHEMBL24257769 0.73 C5AR1 (0.41) SQORGABRG2GABRB3GABRA5GABRA3
SCHEMBL30546869 0.73 C5AR1 (0.41) SQORGABRG2GABRB3GABRA5GABRA3
SCHEMBL24257856 0.73 USP7 (0.43) TP53POLBMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2023-09-21 US disclosed
WO-2022036188-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2022-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE HIF1AN, EGLN3, PHF20 CNR1 4291/4885SQOR 756/4885GABRG2 3174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.