SCHEMBL24257742

SCHEMBL24257742

CCNC(=O)c1ncc(-c2ccc(C)nc2)c(C)c1O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.41
EGLN1 Q9GZT9 7/20 0.41
VEGFA P15692 4/20 0.41
FLT1 P17948 4/20 0.41
EGLN3 Q9H6Z9 2/20 0.41
CNR1 P21554 1/20 0.40
IDO1 P14902 1/20 0.38
ACVR1 Q04771 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CFTR P13569 2/20 0.37
WNT1 P04628 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24257601 0.87 EGLN1 (0.56) EGLN1VEGFAFLT1EGLN3
SCHEMBL30546834 0.87 EGLN1 (0.56) EGLN1VEGFAFLT1EGLN3
SCHEMBL30546836 0.85 EGLN1 (0.58) EGLN1VEGFAFLT1EGLN3
SCHEMBL30452450 0.85 EGLN1 (0.58) EGLN1VEGFAFLT1EGLN3
SCHEMBL24257716 0.85 EGLN1 (0.58) EGLN1VEGFAFLT1EGLN3
SCHEMBL24257711 0.76 GRM4 (0.48) EGLN1KDM4E
SCHEMBL30546862 0.73 EGLN3 (0.55) EGLN1VEGFAFLT1EGLN3
SCHEMBL24257682 0.73 EGLN3 (0.55) EGLN1VEGFAFLT1EGLN3
SCHEMBL30546813 0.73 EGLN1 (0.44) EGLN1VEGFAFLT1EGLN3HDAC6
SCHEMBL30454632 0.73 EGLN1 (0.48) EGLN1VEGFAFLT1EGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022036188-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2022-02-17 WO disclosed