SCHEMBL30454632

SCHEMBL30454632

Cc1ccc2cc(-c3cnc(C(=O)NCC(=O)O)c(O)c3C)ccc2n1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 19/20 0.48
EGLN3 Q9H6Z9 6/20 0.48
FLT1 P17948 4/20 0.48
VEGFA P15692 4/20 0.48
FTO Q9C0B1 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24257501 1.00 EGLN1 (0.48) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL24257795 0.88 EGLN1 (0.41) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL30452729 0.88 EGLN1 (0.41) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL24257637 0.87 EGLN1 (0.50) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL24257567 0.86 EGLN1 (0.65) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL30546834 0.84 EGLN1 (0.56) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL30452349 0.84 AKR1C3 (0.42)
SCHEMBL24257500 0.84 AKR1C3 (0.42)
SCHEMBL24257601 0.84 EGLN1 (0.56) EGLN1EGLN3FLT1VEGFAFTO
SCHEMBL24257636 0.83 EGLN1 (0.51) EGLN1EGLN3FLT1VEGFAFTO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4196466-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE Akebia Therapeutics Inc. (US) 2023-06-21 EP disclosed