SCHEMBL24258239

SCHEMBL24258239

NC(=O)Cc1ccc(CNc2ncnc(N(Cc3ccc(C(F)(F)F)cc3)C3CCC3)c2P)cc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 18/20 0.46
AURKA O14965 17/20 0.46
AURKB Q96GD4 9/20 0.46
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19640438 0.90 RPS6KB1 (0.47) RPS6KB1AURKAAURKBEGFR
SCHEMBL19640477 0.87 RPS6KB1 (0.48) RPS6KB1AURKAAURKBEGFR
SCHEMBL19650854 0.84 RORC (0.41) RPS6KB1AURKAAURKB
SCHEMBL19650845 0.81 RPS6KB1 (0.42) RPS6KB1AURKAAURKB
SCHEMBL19640771 0.80 RPS6KB1 (0.43) RPS6KB1AURKAAURKBEGFR
SCHEMBL29397492 0.80 RPS6KB1 (0.43) RPS6KB1AURKAAURKBEGFR
SCHEMBL17501311 0.79 RPS6KB1 (0.48) RPS6KB1AURKAAURKBEGFR
SCHEMBL19640537 0.79 RPS6KB1 (0.44) RPS6KB1AURKAAURKBEGFR
SCHEMBL19640533 0.78 AURKA (0.42) RPS6KB1AURKAAURKBEGFR
SCHEMBL19640430 0.78 AURKA (0.41) RPS6KB1AURKAAURKBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177612-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2022-02-23 EP disclosed