SCHEMBL24258451

SCHEMBL24258451

CC(F)(F)c1ccc(CN(c2ncnc(NC3CCC4CCC(CCS(C)(=O)=O)CC43)c2F)C2CC2)cc1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.31
CCR5 P51681 1/20 0.31
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19650941 0.83 CACNA1B (0.35) CCR2CCR5JAK2JAK1
SCHEMBL19640694 0.78 CACNA1B (0.37) CCR2CCR5JAK2JAK1
SCHEMBL19650873 0.75 AURKA (0.35) CCR2CCR5
SCHEMBL19650933 0.75 RORC (0.40) JAK2JAK1
SCHEMBL19650849 0.74 RORC (0.39) JAK2JAK1
SCHEMBL24258279 0.73 CACNA1B (0.33)
SCHEMBL19650884 0.72 TRPV1 (0.36)
SCHEMBL19650874 0.72 RORC (0.39) JAK1
SCHEMBL19650885 0.72 RORC (0.37) JAK2JAK1TYK2
SCHEMBL19650872 0.72 RORC (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177612-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2022-02-23 EP disclosed