SCHEMBL2425961

SCHEMBL2425961

COc1ccccc1CNC(=N)Nc1nnc(-c2ccccc2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.56
SMN1; SMN2 Q16637 2/20 0.53
RAB9A P51151 7/20 0.52
GAA P10253 1/20 0.52
CYP2D6 P10635 1/20 0.51
POLB P06746 3/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
CYP2C19 P33261 2/20 0.49
RXFP1 Q9HBX9 2/20 0.47
HTT P42858 1/20 0.47
GLS O94925 1/20 0.47
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MAPT P10636 1/20 0.45
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL2381297 0.96 NPC1 (0.57) NPC1SMN1; SMN2RAB9AGAACYP2D6
SCHEMBL2380611 0.88 NPC1 (0.56) NPC1SMN1; SMN2RAB9AGAAPOLB
SCHEMBL2379377 0.86 SMN1; SMN2 (0.70) NPC1SMN1; SMN2RAB9AGAACYP2D6
SCHEMBL15911601 0.80 MAPT (0.57) NPC1SMN1; SMN2RAB9APOLBMEN1
SCHEMBL2380781 0.80 ROCK2 (0.67) NPC1RAB9AMEN1KMT2AADORA3
SCHEMBL2381223 0.78 KMT2A (0.61) NPC1SMN1; SMN2RAB9ACYP2D6POLB
SCHEMBL2446393 0.78 NPC1 (0.55) NPC1SMN1; SMN2RAB9AGAACYP2D6
SCHEMBL2379500 0.77 NPC1 (0.56) NPC1SMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL2378260 0.76 GAA (0.55) NPC1SMN1; SMN2RAB9AGAAPOLB
Hydrochloric Acid SCHEMBL2381238 0.75 GAA (0.54) NPC1SMN1; SMN2RAB9AGAACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716127-B1 GUANIDINE COMPOUNDS, AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBVIE DEUTSCHLAND (DE) 2014-08-06 EP disclosed
EP-2380885-A1 Guanidine compounds and use of same as binding partners for 5-HT5 receptors Abbott GmbH & Co. KG (DE) 2011-10-26 EP disclosed
EP-2366392-A1 Guanidine compounds and use of same as binding partners for 5-HT5 receptors Abbott GmbH & Co. KG (DE) 2011-09-21 EP disclosed
EP-2366697-A1 Guanidine compounds and use of same as binding partners for 5-HT5 receptors Abbott GmbH & Co. KG (DE) 2011-09-21 EP disclosed