SCHEMBL24259944

SCHEMBL24259944

C/C=C/c1ccc(C2(c3ccc4c(c3)C(C)(C)CCC4(C)C)SCCS2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP26B1 Q9NR63 4/20 0.71
RXRA P19793 10/20 0.60
CYP26A1 O43174 6/20 0.60
CYP3A4 P08684 3/20 0.57
RARB P10826 9/20 0.44
RARG P13631 9/20 0.44
RARA P10276 7/20 0.44
RXRB P28702 4/20 0.39
RXRG P48443 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
GMNN O75496 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17911582 0.83 CYP26B1 (1.00) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL17911581 0.83 CYP26B1 (1.00) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL17914358 0.80 CYP26B1 (0.77) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL8902795 0.78 RARB (0.59) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL8902801 0.78 RARB (0.59) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL24259953 0.78 CYP26B1 (0.71) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL2808583 0.75 RXRA (1.00) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL17911572 0.73 CYP26B1 (1.00) CYP26B1RXRACYP26A1CYP3A4RXRB
SCHEMBL8708782 0.72 RXRA (0.74) CYP26B1RXRACYP26A1CYP3A4RARB
SCHEMBL24259975 0.70 CYP26A1 (0.76) CYP26B1RXRACYP26A1CYP3A4RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3044216-B1 NOVEL AND SPECIFIC INHIBITORS OF CYTOCHROME P450 26 RETINOIC ACID HYDROXYLASE UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2022-02-23 EP disclosed