SCHEMBL2429291

SCHEMBL2429291

O=Cc1csc(B(O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
PTGS2 P35354 1/20 0.31
RAB9A P51151 1/20 0.31
CYP2A6 P11509 1/20 0.31
ALDH5A1 P51649 1/20 0.30
ABAT P80404 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15676434 0.70
SCHEMBL7537600 0.68
SCHEMBL346857 0.67
SCHEMBL152939 0.67
SCHEMBL1503787 0.65
SCHEMBL12422 0.65
SCHEMBL154878 0.65
SCHEMBL8226713 0.65
SCHEMBL4452150 0.65
SCHEMBL1244035 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2026-03-17 US disclosed
WO-2024253416-A1 PYRIMIDINE/PYRIDINE DERIVATIVES OR SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME YUHAN CORPORATION (KR) 2024-12-12 WO disclosed
US-20240166644-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS ASCENTAGE PHARMA GROUP CORP LIMITED (CN) 2024-05-23 US disclosed
CN-114835704-B Sulfonylbenzamide derivatives as BCL-2 inhibitors 苏州亚盛药业有限公司 2023-10-27 CN disclosed
CN-113292540-B N-fluorenyl benzocarbazole compound taking quinoxaline as auxiliary receptor, preparation method and application thereof 浙江工业大学 2023-10-20 CN disclosed
CN-113292540-A N-fluorenyl benzocarbazole compound with quinoxaline as auxiliary receptor, preparation method and application thereof 浙江工业大学 2021-08-24 CN disclosed
EP-2366699-B1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF ASAHI KASEI PHARMA CORP (JP) 2013-08-07 EP disclosed
US-8299055-B2 8-substituted isoquinoline derivative and the use thereof ASAHI KASEI PHARMA CORPORATION (JP) 2012-10-30 US disclosed
EP-2366699-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF Asahi Kasei Pharma Corporation (JP) 2011-09-21 EP disclosed
US-20100261701-A1 8-Substituted isoquinoline derivative and the use thereof ASAHI KASEI PHARMA CORPORATION (JP) 2010-10-14 US disclosed
US-5698574-A BACTERICIDE BAYER AKTIENGESELLSCHAFT (DE) 1997-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors BCL2A1, BCL2L1, BCL2L11 KDM4E 3052/4885PTGS2 2422/4885RAB9A 1139/4885
US-20240166644-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS BCL2, BCL2L2, BCL2L1 KDM4E 1780/4885PTGS2 1531/4885RAB9A 1036/4885
US-20100261701-A1 8-Substituted isoquinoline derivative and the use thereof RELA, NFKBIA, NFKB2 KDM4E 2465/4885PTGS2 270/4885RAB9A 2223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.