SCHEMBL24310893

SCHEMBL24310893

CCC(=O)c1ncn(Cc2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.48
RIPK1 Q13546 12/20 0.46
KLK1 P06870 1/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20095692 0.88 KLKB1 (0.47) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL19658305 0.84 KLKB1 (0.50) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL1414358 0.84 KLKB1 (0.49) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL24311093 0.82 HDAC1 (0.49) HDAC1HDAC6ALDH1A1
SCHEMBL11584045 0.81 KLKB1 (0.50) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL24094026 0.81 KLKB1 (0.59) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL1719033 0.81 ALDH1A1 (0.56) KLKB1RIPK1KLK1ALDH1A1
SCHEMBL1414421 0.81 KLKB1 (0.50) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL18372877 0.81 KLKB1 (0.56) KLKB1RIPK1KLK1HDAC1HDAC6
SCHEMBL1261550 0.79 SMN1; SMN2 (0.41) KLKB1RIPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3978492-A1 BICYCLIC COMPOUND AS RIP-1 KINASE INHIBITOR AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2022-04-06 EP disclosed