SCHEMBL24313200

SCHEMBL24313200

CNC(=O)c1ccc(OC)c(C2COCCCN2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
PLK1 P53350 2/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
PDE4D Q08499 5/20 0.38
PDE4A P27815 4/20 0.38
PDE4B Q07343 4/20 0.38
PDE4C Q08493 4/20 0.38
CLK1 P49759 2/20 0.37
CLK2 P49760 2/20 0.37
GABRA5 P31644 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29456495 0.89 KMT2A (0.43) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL21491449 0.89 KMT2A (0.43) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL21491303 0.87 CA12 (0.44) PDE4DPDE4APDE4BPDE4CMAPT
Hydrochloric Acid SCHEMBL29456315 0.86 CA12 (0.43) PDE4DPDE4APDE4BPDE4CMAPT
Hydrochloric Acid SCHEMBL21491110 0.86 CA12 (0.43) PDE4DPDE4APDE4BPDE4CMAPT
SCHEMBL24313112 0.82 SCN9A (0.39) SLC6A2SLC6A4SLC6A3CLK1CLK2
SCHEMBL21491317 0.75 ALDH1A1 (0.41) SLC6A2SLC6A4SLC6A3KMT2AMEN1
SCHEMBL21491473 0.73 ALDH1A1 (0.39) SLC6A2SLC6A4SLC6A3KMT2AMEN1
SCHEMBL22516364 0.72 MEN1 (0.49) CCNCCDK8PLK1PDE4DPDE4A
SCHEMBL25482905 0.72 TSHR (0.37) KMT2AMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4043460-A1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF Merck Patent GmbH (DE) 2022-08-17 EP disclosed
EP-3784666-B1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2022-03-16 EP disclosed