SCHEMBL24316749

SCHEMBL24316749

COC(=O)c1cnn(Cc2ccc(N3CCC(C)C3)nc2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 5/20 0.61
BTK Q06187 7/20 0.46
RAB9A P51151 6/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPK1 P28482 2/20 0.44
NPC1 O15118 5/20 0.43
HPGD P15428 3/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KLK1 P06870 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.40
GRM2 Q14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18795838 0.89 KLKB1 (0.61) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL18796211 0.89 KLKB1 (0.61) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL24316756 0.89 KLKB1 (0.61) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL20538997 0.88 KLKB1 (0.61) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL20538998 0.88 KLKB1 (0.61) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
Lithium Ion SCHEMBL29536224 0.87 KLKB1 (0.62) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL21953537 0.85 BTK (0.56) KLKB1BTKGRM2
SCHEMBL18823654 0.83 KLKB1 (0.51) KLKB1BTKRAB9ASMN1; SMN2ALDH1A1
SCHEMBL20549564 0.82 BTK (0.59) KLKB1BTKRAB9ANPC1HPGD
SCHEMBL18815404 0.82 BTK (0.59) KLKB1BTKRAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3368529-B1 HETEROARYLCARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2022-04-06 EP disclosed