SCHEMBL24322182

SCHEMBL24322182

Cc1csc2c(C3CC3)n(C)nc12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
PDE4B Q07343 1/20 0.33
PDE7A Q13946 1/20 0.33
GPR35 Q9HC97 1/20 0.33
PDPK1 O15530 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24322357 0.74 PDPK1 (0.38) NPC1PKMPDPK1SMN1; SMN2
SCHEMBL24322356 0.72 PDPK1 (0.36) NPC1PKMPDPK1SMN1; SMN2
SCHEMBL24322139 0.69 PDPK1 (0.34) NPC1PKMPDPK1SMN1; SMN2
SCHEMBL24322198 0.67 PDPK1 (0.36) NPC1PKMGPR35PDPK1SMN1; SMN2
SCHEMBL24322110 0.67 PDPK1 (0.33) NPC1PKMPDPK1SMN1; SMN2
SCHEMBL25235457 0.66 NPC1 (0.32) NPC1PKM
SCHEMBL23519900 0.62 PDE10A (0.50) PDE4BPDE7A
SCHEMBL16132460 0.61 GRM5 (0.33)
SCHEMBL12967352 0.61 MAP4K4 (0.40)
SCHEMBL15269532 0.60 KDM4E (0.36) NPC1SMN1; SMN2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
WO-2022061273-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS, INCORPORATED (US) 2022-03-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals CDK6, CDK1, CDK3 NPC1 3950/4885PKM 410/4885PDE4B 1545/4885
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals CDK6, CDK1, CDK3 NPC1 3950/4885PKM 410/4885PDE4B 1545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.