SCHEMBL24322198

SCHEMBL24322198

CC(=O)c1c2scc(C)c2nn1C

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.36
GPR35 Q9HC97 3/20 0.33
MAPK1 P28482 3/20 0.32
ALDH1A1 P00352 2/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 3/20 0.32
KDM4E B2RXH2 2/20 0.32
RXFP1 Q9HBX9 2/20 0.32
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24322110 0.83 PDPK1 (0.33) PDPK1MAPK1SMN1; SMN2NPC1PKM
SCHEMBL24322357 0.74 PDPK1 (0.38) PDPK1MAPK1SMN1; SMN2NPC1PKM
SCHEMBL24322356 0.72 PDPK1 (0.36) PDPK1MAPK1SMN1; SMN2NPC1PKM
SCHEMBL24322139 0.69 PDPK1 (0.34) PDPK1SMN1; SMN2NPC1PKM
SCHEMBL25233556 0.69 TNKS (0.32) ALDH1A1TNKSPARP1TNKS2
SCHEMBL24322182 0.67 NPC1 (0.35) PDPK1GPR35SMN1; SMN2NPC1PKM
SCHEMBL25235457 0.66 NPC1 (0.32) NPC1PKM
SCHEMBL12647732 0.61 KDM4E (0.42) ALDH1A1SMN1; SMN2PKMMAPTRAB9A
SCHEMBL16433568 0.61 KDM4E (0.42) ALDH1A1SMN1; SMN2MAPTRAB9AKDM4E
SCHEMBL13683180 0.60 KDM4E (0.41) ALDH1A1SMN1; SMN2MAPTRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2023-11-09 US disclosed
CN-116583283-A CDK inhibitors and their use as pharmaceuticals 普莱鲁德疗法有限公司 2023-08-11 CN disclosed
EP-4214213-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS Prelude Therapeutics, Incorporated (US) 2023-07-26 EP disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals PRELUDE THERAPEUTICS INCORPORATED (US) 2023-06-27 US disclosed
WO-2022061273-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS, INCORPORATED (US) 2022-03-24 WO disclosed
WO-2022061273-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS, INCORPORATED (US) 2022-03-24 WO disclosed
US-20220089608-A1 CDK Inhibitors And Their Use As Pharmaceuticals PRELUDE THERAPEUTICS, INCORPORATED 2022-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220089608-A1 CDK Inhibitors And Their Use As Pharmaceuticals CDK6, CDK1, CDK3 PDPK1 143/4885GPR35 2875/4885MAPK1 198/4885
US-20230357265-A1 CDK Inhibitors And Their Use As Pharmaceuticals CDK6, CDK1, CDK3 PDPK1 143/4885GPR35 2875/4885MAPK1 198/4885
US-11685744-B2 CDK inhibitors and their use as pharmaceuticals CDK6, CDK1, CDK3 PDPK1 143/4885GPR35 2875/4885MAPK1 198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.