SCHEMBL24323636

SCHEMBL24323636

CC1(CC(C#N)NCc2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
KDM4E B2RXH2 2/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
CTSC P53634 5/20 0.35
CTSS P25774 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK1 P28482 1/20 0.34
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24019759 0.77 SIGMAR1 (0.47) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL18775067 0.76 SIGMAR1 (0.43) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL24323635 0.75 SIGMAR1 (0.41) SIGMAR1CYP3A4SMN1; SMN2HPGD
SCHEMBL24324590 0.74 SIGMAR1 (0.41) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL9779725 0.74 SIGMAR1 (0.43) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL18775058 0.73 SIGMAR1 (0.40) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL18762581 0.73 SIGMAR1 (0.44) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL9676562 0.72 CYP3A4 (0.44) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL20739382 0.72 SIGMAR1 (0.39) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2
SCHEMBL18762460 0.72 SIGMAR1 (0.39) SIGMAR1KDM4ECYP3A4MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196429-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-12 WO disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed