SCHEMBL24324039

SCHEMBL24324039

Cc1c[nH]c2nc(C=O)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
ADORA2A P29274 4/20 0.36
ADORA1 P30542 4/20 0.36
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
TRIM24 O15164 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ATM Q13315 1/20 0.33
CYP2A6 P11509 1/20 0.31
FGFR4 P22455 1/20 0.30
RRM2 P31350 1/20 0.30
GAA P10253 1/20 0.30
MAPK1 P28482 1/20 0.30
PRMT5 O14744 1/20 0.30
WDR77 Q9BQA1 1/20 0.30
BTK Q06187 1/20 0.30
ITK Q08881 1/20 0.30
PDE4A P27815 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29600275 0.79 CCR1 (0.39) CCR1ADORA2AADORA1KMT2AALDH1A1
SCHEMBL24323860 0.79 CCR1 (0.39) CCR1ADORA2AADORA1KMT2AALDH1A1
SCHEMBL15333269 0.76 CDK5 (0.46) ADORA2AADORA1KMT2AMEN1ALDH1A1
SCHEMBL7922469 0.75 ADORA2A (0.53) ADORA2AADORA1KMT2AMEN1ALDH1A1
SCHEMBL13834371 0.75 LRRK2 (0.49) CCR1PRMT5WDR77
SCHEMBL29956652 0.73 AXL (0.45) MAPK1BTKITK
SCHEMBL21589019 0.72 ADORA2A (0.40) ADORA2AADORA1KMT2AMEN1ALDH1A1
SCHEMBL11467387 0.71 CSNK2A2 (0.48) ADORA2AADORA1KMT2AMEN1ALDH1A1
SCHEMBL6176944 0.68 CCR1 (0.54) CCR1KMT2AMEN1ALDH1A1KDM4E
SCHEMBL24096805 0.68 NR4A2 (0.44) KMT2AMEN1ALDH1A1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed