SCHEMBL24324154

SCHEMBL24324154

Cn1ccc2ccc(C=O)nc21

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.47
CYP2A6 P11509 2/20 0.44
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TRIM24 O15164 1/20 0.35
TRIM33 Q9UPN9 1/20 0.35
FGFR4 P22455 1/20 0.34
BRD4 O60885 1/20 0.31
TAF1 P21675 1/20 0.31
BRPF1 P55201 1/20 0.31
CREBBP Q92793 1/20 0.31
CECR2 Q9BXF3 1/20 0.31
BRD9 Q9H8M2 1/20 0.31
PIK3CB P42338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21284819 0.76 CCR1 (0.45) CCR1ALDH1A1BRD4BRPF1BRD9
SCHEMBL29600465 0.74 DDB1 (0.35) DDB1CRBNALDH1A1
SCHEMBL24323565 0.74 DDB1 (0.35) DDB1CRBNALDH1A1
SCHEMBL7914425 0.71 CCR1 (0.42) CCR1CYP2A6DDB1CRBNBRD4
SCHEMBL30322466 0.69 DDB1 (0.39) CYP2A6DDB1CRBNPIK3CB
SCHEMBL22323347 0.69 DDB1 (0.39) CYP2A6DDB1CRBNPIK3CB
SCHEMBL15091312 0.69 PIK3CB (0.44) CYP2A6DDB1CRBNPIK3CB
SCHEMBL30545112 0.69 DDB1 (0.39) CYP2A6DDB1CRBNPIK3CB
SCHEMBL30503575 0.69 APP (0.42) CYP2A6DDB1CRBNPIK3CB
SCHEMBL3754475 0.69 DDB1 (0.39) CYP2A6DDB1CRBNPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601158-A Modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-08-15 CN disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed