SCHEMBL24326317

SCHEMBL24326317

CN1CCN(Cc2ccccc2)C(CO)C1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.67
MC4R P32245 1/20 0.49
ALDH1A1 P00352 1/20 0.48
POLB P06746 2/20 0.48
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3436828 1.00 SIGMAR1 (0.67) SIGMAR1MC4RALDH1A1POLBGAA
SCHEMBL7383165 0.86 SIGMAR1 (0.60) SIGMAR1MC4RALDH1A1POLB
SCHEMBL4821732 0.84 SIGMAR1 (0.59) SIGMAR1MC4R
SCHEMBL4821722 0.84 SIGMAR1 (0.59) SIGMAR1MC4R
SCHEMBL15829968 0.84 GBA1 (0.53) SIGMAR1ALDH1A1POLB
SCHEMBL25154270 0.84 SIGMAR1 (0.59) SIGMAR1MC4RALDH1A1
SCHEMBL25154734 0.84 SIGMAR1 (0.59) SIGMAR1MC4RALDH1A1
SCHEMBL65364 0.83 SIGMAR1 (0.78) SIGMAR1ALDH1A1POLBGAA
SCHEMBL20719 0.83 SIGMAR1 (0.78) SIGMAR1ALDH1A1POLBGAA
SCHEMBL2974293 0.83 SIGMAR1 (0.78) SIGMAR1ALDH1A1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed