SCHEMBL2432649

SCHEMBL2432649

CCC(C(=O)O)c1cc(OC)c(N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.40
AKR1C2 P52895 8/20 0.40
AKR1C1 Q04828 2/20 0.40
PTGS1 P23219 1/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
RAB9A P51151 2/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 1/20 0.37
USP2 O75604 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CREBBP Q92793 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151815 0.83 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1PTGS1AKR1B10
SCHEMBL2430732 0.79 AKR1C3 (0.38) AKR1C3AKR1C2AKR1C1LMNASMN1; SMN2
SCHEMBL28041376 0.77 AKR1C3 (0.46) AKR1C3AKR1C2AKR1C1PTGS1LMNA
SCHEMBL28041375 0.77 AKR1C3 (0.46) AKR1C3AKR1C2AKR1C1PTGS1LMNA
SCHEMBL30231208 0.76 AKR1C3 (0.44) AKR1C3AKR1C2AKR1C1PTGS1AKR1B10
SCHEMBL536349 0.76 AKR1C3 (0.44) AKR1C3AKR1C2AKR1C1PTGS1AKR1B10
SCHEMBL2412837 0.74 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1PTGS1STING1
SCHEMBL1589867 0.73 AKR1C3 (0.46) AKR1C3AKR1C2AKR1C1PTGS1AKR1B10
SCHEMBL28784595 0.71 MAPT (0.35) AKR1C3AKR1C2LMNAALDH1A1RAB9A
SCHEMBL29889833 0.70 POLB (0.53) AKR1C3AKR1C2AKR1C1PTGS1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed