SCHEMBL2430732

SCHEMBL2430732

CCC(C(=O)O)c1cc(Cl)c(N)cc1F

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.38
AKR1C2 P52895 8/20 0.38
KDM4E B2RXH2 1/20 0.35
AKR1B10 O60218 1/20 0.33
AKR1C4 P17516 1/20 0.33
AKR1C1 Q04828 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151815 0.86 AKR1C3 (0.40) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL2432649 0.79 AKR1C3 (0.40) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL30231208 0.79 AKR1C3 (0.44) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL536349 0.79 AKR1C3 (0.44) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL1589867 0.75 AKR1C3 (0.46) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL13532054 0.75 KMT2A (0.38) KDM4ESMN1; SMN2
SCHEMBL30193006 0.73 AKR1C3 (0.45) AKR1C3AKR1C2AKR1C1
SCHEMBL1590616 0.72 AKR1C3 (0.50) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL16963923 0.71 CES2 (0.46) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL29010117 0.71 KEAP1 (0.47) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed