SCHEMBL24327015

SCHEMBL24327015

Cc1ccc(Nc2nc(Cl)ncc2Cl)c2c1CCN2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 10/20 0.38
CDK2 P24941 10/20 0.38
CDK9 P50750 10/20 0.38
CCNK O75909 9/20 0.38
CCND3 P30281 8/20 0.38
CDK6 Q00534 8/20 0.38
ALK Q9UM73 1/20 0.35
LRRK2 Q5S007 1/20 0.34
MAPK3 P27361 1/20 0.32
MAP4K1 Q92918 1/20 0.32
CDK7 P50613 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29661304 1.00 CCNA2 (0.38) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL29661462 0.85 ALK (0.33) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24327455 0.85 IGF1R (0.35) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24328293 0.85 ALK (0.33) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24327456 0.82 ALK (0.32) ALK
SCHEMBL29661395 0.78 MAP4K1 (0.38) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24327605 0.78 MAP4K1 (0.38) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL29661540 0.76 MAP4K1 (0.35) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24328349 0.76 MAP4K1 (0.35) CCNA2CDK2CDK9CCNKCCND3
SCHEMBL24327586 0.73 IGF1R (0.35) CCNA2CDK2CDK9CCNKCCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
CN-116249690-A Indoline compounds and derivatives as EGFR inhibitors 百济神州有限公司 2023-06-09 CN disclosed
WO-2022063106-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEIGENE, LTD. (KY) 2022-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS EGFR, ERBB2, ERBB4 CCNA2 1420/4885CDK2 42/4885CDK9 67/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.