SCHEMBL24328340

SCHEMBL24328340

Cc1cc2c(c(Nc3nc(Cl)ncc3Cl)c1)N(S(C)(=O)=O)CC2

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 12/20 0.38
AXL P30530 2/20 0.38
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37
MET P08581 3/20 0.35
EGFR P00533 1/20 0.34
CHEK1 O14757 1/20 0.34
KIT P10721 1/20 0.34
FLT3 P36888 1/20 0.34
INSR P06213 1/20 0.34
MAPK3 P27361 1/20 0.33
CCND3 P30281 1/20 0.33
CDK6 Q00534 1/20 0.33
MAP4K1 Q92918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29661327 1.00 ALK (0.38) ALKAXLCDK7CDK9MET
SCHEMBL24327468 0.84 CDK9 (0.43) ALKAXLCDK7CDK9MET
SCHEMBL29661342 0.84 CDK9 (0.43) ALKAXLCDK7CDK9MET
SCHEMBL29661357 0.79 ALK (0.42) ALKCDK7CDK9EGFRMAPK3
SCHEMBL24327449 0.79 ALK (0.42) ALKCDK7CDK9EGFRMAPK3
SCHEMBL29661271 0.78 CDK9 (0.42) ALKAXLCDK7CDK9MET
SCHEMBL26778572 0.78 CDK9 (0.42) ALKAXLCDK7CDK9MET
SCHEMBL24327587 0.77 BRD4 (0.37) CDK7CDK9CCND3CDK6
SCHEMBL29661472 0.77 BRD4 (0.37) CDK7CDK9CCND3CDK6
SCHEMBL24327597 0.76 ALK (0.41) ALKCDK7CDK9EGFRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEONE MEDICINES I GMBH (CH) 2023-11-23 US disclosed
WO-2022063106-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEIGENE, LTD. (KY) 2022-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230373960-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS EGFR, ERBB2, ERBB4 ALK 13/4885AXL 81/4885CDK7 216/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.