SCHEMBL24328554

SCHEMBL24328554

BC1(B)Oc2cc3ncnc(Nc4cccc(Br)c4F)c3cc2OC1(B)B

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.72
RET P07949 1/20 0.46
KIF5B P33176 1/20 0.46
KDR P35968 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20865336 0.86 EGFR (0.72) EGFRKDR
SCHEMBL20865211 0.84 EGFR (1.00) EGFR
SCHEMBL29363644 0.84 EGFR (1.00) EGFR
SCHEMBL24329506 0.84 EGFR (0.87) EGFRKDR
SCHEMBL31004070 0.84 EGFR (1.00) EGFR
SCHEMBL20865222 0.82 EGFR (0.72) EGFRRETKIF5BKDR
SCHEMBL20856929 0.82 EGFR (0.72) EGFRRETKIF5BKDR
SCHEMBL24329439 0.82 EGFR (0.91) EGFR
SCHEMBL20865245 0.82 EGFR (0.72) EGFRRETKIF5BKDR
SCHEMBL29394159 0.82 EGFR (0.72) EGFRRETKIF5BKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024081447-A1 EGFR INHIBITORS FOR TREATING LUNG CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-04-18 WO disclosed
US-20230364091-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-11-16 US disclosed
US-20230358726-A1 NON-INVASIVE FUNCTIONAL COMPANION ASSAYS FOR ONCOGENE TARGETED THERAPY FOR BRAIN CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-11-09 US disclosed
US-11377451-B2 Compositions and methods for treating cancer THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-07-05 US disclosed
WO-2022061202-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-03-24 WO disclosed
US-20220064177-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-03-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11377451-B2 Compositions and methods for treating cancer TP53, EGFR, SLC2A1 EGFR 2/4885RET 214/4885KIF5B 934/4885
US-20230364091-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TP53, EGFR, SLC2A1 EGFR 2/4885RET 221/4885KIF5B 1293/4885
US-20220064177-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TP53, SLC2A1, EGFR EGFR 3/4885RET 262/4885KIF5B 1221/4885
US-20230358726-A1 NON-INVASIVE FUNCTIONAL COMPANION ASSAYS FOR ONCOGENE TARGETED THERAPY FOR BRAIN CANCER EGFR, IDH1, KRAS EGFR 1/4885RET 31/4885KIF5B 1337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.