SCHEMBL2433581

SCHEMBL2433581

COCC(OC1CCC(C)(C(=O)O)CC1)(C(=O)Cc1cc(Cl)c(NC(=O)c2cn(C)c3ccccc23)cc1F)N1CCCC1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 12/20 0.53
ITGA4 P13612 12/20 0.53
KDM1A O60341 1/20 0.36
ACKR3 P25106 1/20 0.35
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
CNR2 P34972 2/20 0.34
S1PR2 O95136 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2429881 0.91 ITGB1 (0.65) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2429858 0.90 ITGB1 (0.55) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2432479 0.89 ITGB1 (0.58) ITGB1ITGA4KDM1AACKR3CNR2
SCHEMBL7265189 0.85 ITGB1 (0.52) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2432754 0.80 ITGB1 (0.66) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2433484 0.80 ITGB1 (0.68) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2433487 0.80 ITGB1 (0.68) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2431891 0.80 ITGB1 (0.68) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL71313 0.80 ITGB1 (0.64) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL71314 0.80 ITGB1 (0.64) ITGB1ITGA4KDM1AACKR3BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed