SCHEMBL7265189

SCHEMBL7265189

CN(C)C(=O)COC(OC1CCC(C)(C(=O)O)CC1)(C(=O)Cc1cc(Cl)c(NC(=O)c2cn(C)c3ccccc23)cc1F)N1CCCC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.52
ITGA4 P13612 13/20 0.52
KDM1A O60341 1/20 0.34
ACKR3 P25106 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2431848 0.92 ITGB1 (0.62) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2434375 0.90 ITGB1 (0.55) ITGB1ITGA4KDM1AACKR3MEN1
SCHEMBL2429858 0.87 ITGB1 (0.55) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2433581 0.85 ITGB1 (0.53) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2437236 0.83 ITGB1 (0.64) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2437230 0.83 ITGB1 (0.64) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2432754 0.83 ITGB1 (0.66) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2434421 0.83 ITGB1 (0.66) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2434426 0.83 ITGB1 (0.66) ITGB1ITGA4KDM1AACKR3BCHE
SCHEMBL2435061 0.82 ITGB1 (0.62) ITGB1ITGA4KDM1AACKR3BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-A1 VLA-4 INHIBITORS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-09-24 EP disclosed