SCHEMBL2434320

SCHEMBL2434320

CC(C(=O)O)c1ccc2nc(-c3cn(C)c4ccccc34)oc2c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.47
ITGA4 P13612 3/20 0.47
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 4/20 0.45
HPGD P15428 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MGAM O43451 2/20 0.41
GAA P10253 2/20 0.41
SI P14410 2/20 0.41
MGAM2 Q2M2H8 2/20 0.41
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2437936 0.89 ITGB1 (0.49) ITGB1ITGA4KDM4EALDH1A1CDK9
SCHEMBL2430872 0.81 ITGB1 (0.58) ITGB1ITGA4KDM4EALDH1A1HPGD
SCHEMBL2429595 0.77 ITGB1 (0.56) ITGB1ITGA4KDM4EALDH1A1HPGD
SCHEMBL2434007 0.74 NPC1 (0.44) ITGB1ITGA4KDM4EALDH1A1HPGD
SCHEMBL2430981 0.71 ITGB1 (0.49) ITGB1ITGA4KDM4EALDH1A1CDK9
SCHEMBL14591811 0.71 ITGB1 (0.50) ITGB1ITGA4CYP3A4CDK2
SCHEMBL2687045 0.71 KDM4E (0.64) KDM4EALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL2435546 0.71 ITGB1 (0.48) ITGB1ITGA4
SCHEMBL2432757 0.71 ITGB1 (0.61) ITGB1ITGA4KDM4EALDH1A1CDK9
SCHEMBL14591814 0.70 ITGB1 (0.45) ITGB1ITGA4KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed