SCHEMBL2435546

SCHEMBL2435546

CC(C(=O)O)c1ccc2nc(-c3cn(C)c4cc(F)ccc34)oc2c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.48
ITGA4 P13612 5/20 0.48
MAOA P21397 1/20 0.42
ADRA1A P35348 1/20 0.42
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
MET P08581 3/20 0.38
AKR1C3 P42330 4/20 0.37
AKR1C2 P52895 4/20 0.37
HDAC6 Q9UBN7 2/20 0.35
FASN P49327 1/20 0.35
UTRN P46939 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430981 0.93 ITGB1 (0.49) ITGB1ITGA4MAOAADRA1AMET
SCHEMBL2435828 0.83 MAOA (0.53) ITGB1ITGA4MAOAADRA1AMET
SCHEMBL2433950 0.81 ITGB1 (0.59) ITGB1ITGA4IDO1TDO2MET
SCHEMBL14591805 0.81 ITGB1 (0.55) ITGB1ITGA4IDO1TDO2MET
SCHEMBL2433361 0.79 ITGB1 (0.47) ITGB1ITGA4MAOAADRA1AAKR1C3
SCHEMBL14626706 0.79 ITGB1 (0.57) ITGB1ITGA4IDO1TDO2MET
SCHEMBL14592396 0.77 ITGB1 (0.57) ITGB1ITGA4IDO1TDO2MET
SCHEMBL12327757 0.77 ITGB1 (0.51) ITGB1ITGA4IDO1TDO2MET
SCHEMBL2437936 0.77 ITGB1 (0.49) ITGB1ITGA4MET
SCHEMBL2434541 0.75 ITGB1 (0.60) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed