Fentiazac

Fentiazac

SCHEMBL24355

O=C(O)Cc1sc(-c2ccccc2)nc1-c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 17/20 1.00
KDM4E B2RXH2 4/20 1.00
ALDH1A1 P00352 3/20 1.00
CYP1A2 P05177 1/20 1.00
CYP2C9 P11712 1/20 1.00
HPGD P15428 1/20 1.00
CYP2C19 P33261 1/20 1.00
POLB P06746 1/20 0.83
MEN1 O00255 1/20 0.71
MAPT P10636 1/20 0.71
KMT2A Q03164 1/20 0.71
SMN1; SMN2 Q16637 1/20 0.71
RXFP1 Q9HBX9 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fentiazac SCHEMBL16196751 1.00 PTGDR2 (1.00) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL1514667 1.00 PTGDR2 (1.00) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
Fentiazac SCHEMBL5390943 0.99 PTGDR2 (0.97) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL4497493 0.91 PTGDR2 (1.00) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL11100736 0.90 PTGDR2 (0.82) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL13116312 0.89 PTGDR2 (0.81) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL12608906 0.89 PTGDR2 (0.81) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL5210404 0.86 PTGDR2 (0.76) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL2818129 0.86 PTGDR2 (1.00) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL13116322 0.85 PTGDR2 (0.74) PTGDR2KDM4EALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 17390 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4662203-A1 BINDARIT CONJUGATES, COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES OR DISORDERS Translatum Medicus Inc. (CA) 2025-12-17 EP claimed
US-20250041208-A1 NEW INJECTABLE COMBINATION FORMULATION NANEXA AB (SE) 2025-02-06 US claimed
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
EP-4444277-A1 NEW INJECTABLE COMBINATION FORMULATION Nanexa AB (SE) 2024-10-16 EP claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
US-20240299348-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE CARAWAY THERAPEUTICS, INC. 2024-09-12 US claimed
WO-2024165925-A1 BINDARIT CONJUGATES, COMPOSITIONS AND METHODS FOR TREATING OCULAR DISEASES OR DISORDERS Translatum Medicus Inc. (CA) 2024-08-15 WO claimed
EP-4398874-A1 INJECTABLE HIGH CONCENTRATION PHARMACEUTICAL FORMULATIONS AND METHODS OF MANUFACTURING AND USE THEREOF Xeris Pharmaceuticals, Inc. (US) 2024-07-17 EP claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-1986003681-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE ABRAHAM 1986-07-03 WO claimed
EP-0180597-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS. SUNSHINE ABRAHAM (US) 1986-05-14 EP claimed
WO-1985004589-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS SUNSHINE ABRAHAM 1985-10-24 WO claimed
US-4545992-A ANTINFLAMMATORY AGENTS, ANALGESICS TOKO YAKUHIN INDUSTRY CO., LTD. (JP) 1985-10-08 US claimed
WO-1985003443-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING DIPHENHYDRAMINE AND METHODS OF USING SAME RICHARDSON-VICKS, INC. (US) 1985-08-15 WO claimed
EP-0114886-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE. SUNSHINE ABRAHAM (US) 1984-08-08 EP claimed
US-4455146-A THERMOPLASTIC ELASTOMERS, OILS OR FATTY ACID, TACKFIER, AND A MEDICINE HISAMITSU PHARMACEUTICAL CO., LTD. (JP) 1984-06-19 US claimed
WO-1984000490-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE AND METHODS OF USING SAME SUNSHINE ABRAHAM 1984-02-16 WO claimed
EP-0072462-A2 Pharmaceutical preparations Toko Yakuhin Industry Co., Ltd. (JP) 1983-02-23 EP claimed
US-4127663-A Thiazole derivatives to treat inflammation JOHN WYETH & BROTHER LIMITED (GB) 1978-11-28 US claimed