SCHEMBL2436747

SCHEMBL2436747

CNC(=O)c1c(-c2ccc(F)cc2)oc2cccc(F)c12

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.45
KCNH2 Q12809 6/20 0.44
CYP2C8 P10632 3/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
CYP3A4 P08684 2/20 0.42
CACNA1C Q13936 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18038612 0.83 KCNH2 (0.43) KCNH2CYP2C8KDM4EALDH1A1HPGD
SCHEMBL6120196 0.83 CYP3A4 (0.48) KCNH2CYP2C8CYP3A4
SCHEMBL1919191 0.82 L3MBTL1 (0.53) KCNH2CYP2C8CYP3A4
SCHEMBL19197887 0.80 KCNH2 (0.50) KCNH2CYP2C8CYP3A4
SCHEMBL1918982 0.80 KCNH2 (0.52) KCNH2CYP2C8
SCHEMBL2368951 0.79 KCNH2 (0.41) KCNH2CYP2C8KDM4ENPC1ALDH1A1
SCHEMBL17464345 0.78 ANO1 (0.42) KCNH2CYP2C8CYP3A4
SCHEMBL2842305 0.77 CYP3A4 (0.54) KCNH2CYP2C8CYP3A4
SCHEMBL17466573 0.76 KCNH2 (0.49) KCNH2CYP2C8CYP3A4
SCHEMBL19198543 0.76 KCNH2 (0.41) KCNH2CYP2C8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP claimed
WO-2011112769-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO claimed