SCHEMBL2436952

SCHEMBL2436952

CNC(=O)c1c(-c2ccc(F)cc2)oc2ccc(-c3cccc(C(=O)N(c4ccccn4)C4CC4)c3)nc12

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
CYP2C8 P10632 3/20 0.42
KCNH2 Q12809 3/20 0.42
CYP3A4 P08684 2/20 0.41
NR1I2 O75469 1/20 0.41
CACNA1C Q13936 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936918 0.90 CYP2C8 (0.52) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL2431623 0.87 ALDH1A1 (0.45) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1917571 0.82 CYP3A4 (0.51) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1917701 0.80 CYP3A4 (0.55) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1918435 0.80 CYP2C8 (0.65) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1918592 0.80 CYP2C8 (0.56) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL2431373 0.80 CACNA1C (0.44) CYP2C8KCNH2CYP3A4CACNA1C
SCHEMBL1919040 0.79 CYP2C8 (0.55) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1919264 0.79 CYP2C8 (0.55) ALDH1A1CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL1937027 0.79 CYP2C8 (0.66) CYP2C8KCNH2CYP3A4NR1I2CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed