SCHEMBL24371887

SCHEMBL24371887

CC(=O)NS(=O)(=O)c1ccc(NC(=O)Cc2ccc(Br)c(Oc3cc(Cl)cc(C#N)c3)c2F)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.40
CA2 P00918 10/20 0.40
CA9 Q16790 6/20 0.40
CA12 O43570 5/20 0.40
CYP3A4 P08684 3/20 0.38
SLC22A12 Q96S37 1/20 0.36
RORC P51449 3/20 0.35
CA5A P35218 2/20 0.35
CA7 P43166 2/20 0.35
CA5B Q9Y2D0 2/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
PDK1 Q15118 2/20 0.33
PDK2 Q15119 2/20 0.33
PDK3 Q15120 2/20 0.33
PDK4 Q16654 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Elsulfavirine SCHEMBL1344216 0.93 CA1 (0.40) CA1CA2CA9CA12CYP3A4
Elsulfavirine SCHEMBL1341521 0.93 CA1 (0.40) CA1CA2CA9CA12CYP3A4
Elsulfavirine SCHEMBL1344214 0.93 CA1 (0.39) CA1CA2CA9CA12CYP3A4
Depulfavirine SCHEMBL29421868 0.90 CA1 (0.52) CA1CA2CA9CA12CA5A
Depulfavirine SCHEMBL2638090 0.90 CA1 (0.52) CA1CA2CA9CA12CA5A
SCHEMBL2638424 0.86 CYP3A4 (0.43) CA1CA2CA9CA12CYP3A4
SCHEMBL3833407 0.86 CYP3A4 (0.42) CA1CA2CA9CA12CYP3A4
Elsulfavirine Sodium SCHEMBL29421854 0.85 CA1 (0.38) CA1CA2CA9CA12CYP3A4
Elsulfavirine Sodium SCHEMBL29425195 0.85 CA1 (0.38) CA1CA2CA9CA12CYP3A4
SCHEMBL2639193 0.85 CYP3A4 (0.42) CA1CA2CA9CA12CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3988539-A1 ACTIVE INGREDIENT, PHARMACEUTICAL COMPOSITION, AND MEDICINAL PREPARATION FOR THERAPY OF HIV AND AIDS Alla Chem, LLC (US) 2022-04-27 EP disclosed