SCHEMBL24378028

SCHEMBL24378028

CCS(=O)(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.57
CYP21A2 P08686 3/20 0.57
CYP11B1 P15538 3/20 0.57
CYP3A4 P08684 2/20 0.57
CYP19A1 P11511 1/20 0.57
KDM4E B2RXH2 5/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
CYP2C19 P33261 3/20 0.54
TSHR P16473 2/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 2/20 0.54
CHKA P35790 1/20 0.52
CYP2C9 P11712 2/20 0.49
HIF1A Q16665 2/20 0.49
HSD17B10 Q99714 2/20 0.49
MAPK1 P28482 1/20 0.47
ADRB2 P07550 1/20 0.47
NCF1 P14598 1/20 0.47
PLD1 Q13393 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634850 0.81 KMT2A (0.64) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL1487309 0.81 CHKA (0.55) CYP3A4MAPTCYP2C19TSHRCYP1A2
SCHEMBL12082286 0.80 KMT2A (0.67) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL4142494 0.79 KDM4E (0.55) CYP17A1CYP21A2CYP11B1CYP3A4CYP19A1
SCHEMBL21484324 0.79 KDM4E (0.59) CYP17A1CYP21A2CYP11B1CYP3A4CYP19A1
SCHEMBL763179 0.79 KDM4E (0.59) CYP17A1CYP21A2CYP11B1KDM4EALDH1A1
SCHEMBL27571160 0.79 ALDH1A1 (0.63) CYP17A1CYP21A2CYP11B1CYP3A4CYP19A1
SCHEMBL900049 0.79 MAPT (0.61) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL28112415 0.78 CHKA (0.80) CYP3A4KDM4EMAPTCYP2C19TSHR
SCHEMBL14923965 0.76 KDM4E (0.56) CYP3A4KDM4EALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed