SCHEMBL24401545

SCHEMBL24401545

CCOC(=O)c1cn2c(O)cc(OC)nc2n1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
DPP4 P27487 1/20 0.43
DPP8 Q6V1X1 1/20 0.43
DPP9 Q86TI2 1/20 0.43
POLB P06746 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 1/20 0.41
GABRA2 P47869 4/20 0.40
GABRB2 P47870 4/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18990504 0.80 GAA (0.54) GAAKDM4EALDH1A1HPGDPOLB
SCHEMBL18990153 0.76 GAA (0.53) GAAKDM4EDPP4DPP8DPP9
SCHEMBL27242011 0.75 GAA (0.55) GAAKDM4EALDH1A1HPGDDPP4
SCHEMBL5439236 0.73 GAA (0.52) GAAKDM4EALDH1A1HPGDDPP4
SCHEMBL24378550 0.73 DPP4 (0.53) GAAKDM4EALDH1A1HPGDDPP4
SCHEMBL10469595 0.73
SCHEMBL24401546 0.73 DPP4 (0.44) KDM4EALDH1A1HPGDDPP4DPP8
SCHEMBL24378545 0.71 GAA (0.47) GAAKDM4EALDH1A1HPGDPOLB
SCHEMBL9679460 0.70 CYP1A2 (0.43) GAAKDM4EALDH1A1HPGDPOLB
SCHEMBL14633861 0.69 KDM4E (0.64) GAAKDM4EALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230148450-A9 BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF Revolution Medicines, Inc. 2023-05-11 US disclosed
US-20230148450-A9 BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF Revolution Medicines, Inc. 2023-05-11 US disclosed
US-20220135584-A1 BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF REVOLUTION MEDICINES INC (US) 2022-05-05 US disclosed
CN-113767100-A Bicyclic heteroaryl compounds and uses thereof 锐新医药公司 2021-12-07 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220135584-A1 BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF SOST, SOS1, SOS2 GAA 990/4885KDM4E 4659/4885ALDH1A1 3594/4885
US-20230148450-A9 BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF SOST, SOS1, SOS2 GAA 990/4885KDM4E 4659/4885ALDH1A1 3594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.