SCHEMBL24427232

SCHEMBL24427232

CC(C)(C)OC(=O)Nc1ccc(C(=O)CBr)c(F)n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.36
SCN9A Q15858 4/20 0.36
CYP17A1 P05093 3/20 0.36
ATR Q13535 1/20 0.36
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
METAP1 P53582 1/20 0.34
GRIN2B Q13224 1/20 0.34
BCHE P06276 1/20 0.33
APLNR P35414 1/20 0.33
LCK P06239 1/20 0.33
SYK P43405 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29862857 1.00 AKT1 (0.36) AKT1SCN9ACYP17A1ATRGSK3B
SCHEMBL24427691 0.85 RXFP1 (0.35) AKT1SCN9ACYP17A1ATRGSK3B
SCHEMBL15060517 0.84 ATR (0.39) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL19205217 0.84 ATR (0.39) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL38661717 0.83 ATR (0.49) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL38663529 0.83 ATR (0.49) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL18153003 0.81 MAPK8 (0.42) SCN9AMAPK14
SCHEMBL24427294 0.81 PRMT1 (0.38) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL24726041 0.80 KCNQ3 (0.38) SCN9ACYP17A1ATRGSK3BDYRK1A
SCHEMBL29862959 0.80 KCNQ3 (0.38) SCN9ACYP17A1ATRGSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3998263-A1 TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jemincare Pharmaceuticals Co., Ltd. (CN) 2022-05-18 EP disclosed