SCHEMBL24439409

SCHEMBL24439409

Cc1nc(-c2sc(Cl)cc2COC(=O)N(C)Cc2ccccc2)ncc1O[C@H]1CCC[C@H](C(=O)O)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLCO1B1 Q9Y6L6 8/20 0.43
LPAR1 Q92633 7/20 0.43
ABCB11 O95342 3/20 0.43
ABCC3 O15438 2/20 0.43
ABCC4 O15439 2/20 0.43
SLCO1B3 Q9NPD5 2/20 0.43
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
UBE2N P61088 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24439483 0.94 SLCO1B1 (0.38) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL29517335 0.94 SLCO1B1 (0.38) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL24439604 0.91 KLKB1 (0.37) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL29672289 0.90 SLCO1B1 (0.52) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL29672239 0.90 SLCO1B1 (0.52) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL24439408 0.90 SLCO1B1 (0.52) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL24439488 0.90 SLCO1B1 (0.52) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL24439318 0.89 SLCO1B1 (0.45) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL24439612 0.89 SLCO1B1 (0.51) SLCO1B1LPAR1ABCB11ABCC3ABCC4
SCHEMBL29672276 0.89 SLCO1B1 (0.51) SLCO1B1LPAR1ABCB11ABCC3ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed