SCHEMBL24451

SCHEMBL24451

COc1cccc(-c2ccc(C(=O)c3cccc(O)c3)s2)c1

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 19/20 0.80
HSD17B2 P37059 18/20 0.80
HDAC6 Q9UBN7 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23779 0.92 HSD17B2 (0.67) HSD17B1HSD17B2HDAC6
SCHEMBL23202 0.90 HSD17B2 (0.70) HSD17B1HSD17B2
SCHEMBL30843 0.90 HSD17B2 (0.75) HSD17B1HSD17B2
SCHEMBL23010 0.88 HSD17B1 (0.70) HSD17B1HSD17B2
SCHEMBL22549 0.88 HSD17B2 (0.70) HSD17B1HSD17B2
SCHEMBL18195278 0.87 HSD17B2 (0.65) HSD17B1HSD17B2HDAC6
SCHEMBL22914 0.87 HSD17B1 (0.78) HSD17B1HSD17B2
SCHEMBL24263 0.87 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL23361 0.86 HDAC6 (0.66) HSD17B1HSD17B2HDAC6
SCHEMBL23125 0.84 HSD17B2 (0.65) HSD17B1HSD17B2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed