SCHEMBL24460271

SCHEMBL24460271

CC(C)Oc1ccc(-c2cnc3ccc(-c4ccc(C(C)(C)C)cc4)cn23)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.42
SCN5A Q14524 3/20 0.42
CYP1A2 P05177 1/20 0.41
PIK3CA P42336 1/20 0.41
MTOR P42345 1/20 0.41
PTPN5 P54829 1/20 0.40
RIPK2 O43353 2/20 0.40
PTGES O14684 1/20 0.40
KCNH2 Q12809 1/20 0.40
FLT3 P36888 5/20 0.39
FYN P06241 1/20 0.39
DYRK1A Q13627 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
CYP3A4 P08684 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24460322 1.00 CLK1 (0.42) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781539 0.91 CLK1 (0.47) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781610 0.91 CLK1 (0.43) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781173 0.91 CLK1 (0.43) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781179 0.88 SCN5A (0.46) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781811 0.88 SCN5A (0.46) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL24460329 0.86 PIK3CA (0.42) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL24460263 0.86 KCNH2 (0.43) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781168 0.85 SCN5A (0.50) CLK1SCN5ACYP1A2PIK3CAMTOR
SCHEMBL19781776 0.85 FYN (0.54) CLK1CYP1A2PIK3CAMTORRIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
WO-2022108849-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2022-05-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS C3AR1, C9, C1R CLK1 3537/4885SCN5A 4401/4885CYP1A2 276/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.