SCHEMBL24466337

SCHEMBL24466337

O=C1NCc2c1ccnc2I

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.46
DYRK1A Q13627 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
PIM1 P11309 1/20 0.46
CSNK1A1 P48729 1/20 0.46
ROCK1 Q13464 1/20 0.46
LRRK2 Q5S007 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
LTK P29376 1/20 0.40
MST1R Q04912 1/20 0.40
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
PARP10 Q53GL7 7/20 0.36
PARP11 Q9NR21 7/20 0.36
PRKCI P41743 1/20 0.36
PARP1 P09874 3/20 0.36
ACHE P22303 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31264207 0.77 CDK5 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL30842095 0.77 CDK5 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL15566157 0.77 CLK4 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL16921409 0.77 CDK5 (0.46) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL19984500 0.73 CDK5 (0.42) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL30700995 0.72 CDC7 (0.50) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL1335497 0.71 DYRK1A (0.61) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL30233027 0.69 DYRK1A (0.39) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL21990680 0.68 L3MBTL1 (0.41) CDK5DYRK1ACLK4PIM1CSNK1A1
SCHEMBL30913134 0.68 PRKD1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4005638-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2022-06-01 EP disclosed