SCHEMBL24468673

SCHEMBL24468673

CC(F)(F)CN(Cc1ccc(C(F)(F)F)cn1)C(=O)c1ccc2nc(N)c3c(c2c1)COC3

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.47
WDR77 Q9BQA1 1/20 0.47
TRPM8 Q7Z2W7 2/20 0.37
MCHR1 Q99705 4/20 0.35
SCN9A Q15858 6/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
BCHE P06276 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
CSF1R P07333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24468572 0.95 PRMT5 (0.48) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL29685440 0.95 PRMT5 (0.48) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL27181538 0.93 PRMT5 (0.46) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL24468560 0.92 PRMT5 (0.48) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL29685302 0.92 PRMT5 (0.48) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL27181245 0.90 PRMT5 (0.48) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL24468483 0.89 PRMT5 (0.46) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL29685297 0.89 PRMT5 (0.46) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL24468675 0.89 PRMT5 (0.45) PRMT5WDR77TRPM8MCHR1SCN9A
SCHEMBL29685483 0.89 PRMT5 (0.49) PRMT5WDR77TRPM8MCHR1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115377-A1 TRICYCLIC CARBOXAMIDE DERIVATIVES AS PRMT5 INHIBITORS AMGEN INC. (US) 2022-06-02 WO disclosed