SCHEMBL24469488

SCHEMBL24469488

Nc1cccc2c1C(=O)N(C1CN3CCC1CC3)C2

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 3/20 0.52
CRBN Q96SW2 1/20 0.51
HTR3B O95264 1/20 0.48
ADRA2A P08913 1/20 0.48
KCNE1 P15382 1/20 0.48
ADRA2C P18825 1/20 0.48
CHRM3 P20309 1/20 0.48
SLC6A4 P31645 1/20 0.48
ADRA1A P35348 1/20 0.48
HRH1 P35367 1/20 0.48
DRD3 P35462 1/20 0.48
CHRNA4 P43681 1/20 0.48
KCNQ1 P51787 1/20 0.48
KCNH2 Q12809 1/20 0.48
SCN5A Q14524 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24469672 1.00 HTR3A (0.52) HTR3ACRBNHTR3BADRA2AKCNE1
SCHEMBL4074347 0.84 HTR3A (0.52) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL4087446 0.82 HTR3A (0.56) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL29607124 0.80 HTR3A (0.48) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL4074754 0.79 HTR3A (0.53) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL12714378 0.78 CRBN (0.53) CRBN
SCHEMBL12714376 0.78 CRBN (0.53) CRBN
SCHEMBL6575375 0.78 HTR3A (0.48) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL6575344 0.78 HTR3A (0.48) HTR3AHTR3BADRA2AKCNE1ADRA2C
SCHEMBL6575349 0.78 HTR3A (0.48) HTR3AHTR3BADRA2AKCNE1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115301-A1 MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2022-06-02 WO disclosed