SCHEMBL2447162

SCHEMBL2447162

CC(C)(C)[C@@](C)(Cc1ccccc1)NC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
RECQL P46063 2/20 0.47
CYP1A2 P05177 2/20 0.47
MMP8 P22894 4/20 0.46
MAPK1 P28482 1/20 0.46
CYP2D6 P10635 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
SLC6A2 P23975 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
RIPK1 Q13546 1/20 0.41
TRPA1 O75762 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5948337 0.81 CYP3A4 (0.67) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL4073210 0.77 CYP3A4 (0.46) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL1273081 0.77 CYP3A4 (0.46) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL16162058 0.76 CYP3A4 (0.49) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL4025551 0.76 CYP3A4 (0.49) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL4583207 0.76 CYP3A4 (0.50) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL1273122 0.76 CYP3A4 (0.49) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL3595349 0.75 CYP3A4 (0.51) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL4027524 0.75 CYP3A4 (0.53) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL
SCHEMBL2025506 0.75 CYP3A4 (0.47) CYP3A4ALDH1A1CYP2C9CYP2C19RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed