SCHEMBL24477385

SCHEMBL24477385

CCc1c([C@H](C)CC)nc2[nH]c3ccccc3n2c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.51
ALDH1A1 P00352 5/20 0.51
HPGD P15428 4/20 0.51
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
POLB P06746 2/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
RPA1 P27694 1/20 0.43
PDE2A O00408 1/20 0.43
PDE6D O43924 1/20 0.43
PDE8A O60658 1/20 0.43
PDE5A O76074 1/20 0.43
PDE9A O76083 1/20 0.43
PDE8B O95263 1/20 0.43
PDE6A P16499 1/20 0.43
PDE6G P18545 1/20 0.43
PDE4A P27815 1/20 0.43
PDE6B P35913 1/20 0.43
PDE6C P51160 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24477379 1.00 KDM4E (0.51) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24477393 1.00 KDM4E (0.51) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL29567821 0.93 KDM4E (0.49) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL29567701 0.93 KDM4E (0.49) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL29567688 0.93 KDM4E (0.49) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL23295672 0.91 KDM4E (0.54) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24477380 0.91 KMT2A (0.44) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24477384 0.91 KMT2A (0.44) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24477378 0.91 RAB9A (0.46) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24477398 0.91 KMT2A (0.44) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022111473-A1 COMPOUNDS AS MRGPRX2 ANTAGONISTS BIOARDIS LLC (US) 2022-06-02 WO disclosed
WO-2022111473-A1 COMPOUNDS AS MRGPRX2 ANTAGONISTS BIOARDIS LLC (US) 2022-06-02 WO disclosed