SCHEMBL24528596

SCHEMBL24528596

CN(C)CCC/N=C/c1ccc(-n2ccc3c(-c4ccccc4)nc(-c4ccccc4)nc32)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
MAPK1 P28482 1/20 0.34
THRB P10828 1/20 0.32
NPY1R P25929 1/20 0.32
NPY2R P49146 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ATM Q13315 1/20 0.32
KMT2A Q03164 3/20 0.32
TLR9 Q9NR96 2/20 0.32
MEN1 O00255 2/20 0.32
PSMD14 O00487 1/20 0.32
ACP1 P24666 1/20 0.31
RAD52 P43351 1/20 0.31
POLB P06746 2/20 0.31
HTR7 P34969 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29681045 1.00 KDM4E (0.37) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL24528655 0.96 KDM4E (0.34) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL24528512 0.96 KDM4E (0.37) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL29680746 0.96 KDM4E (0.37) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL24528599 0.95 KDM4E (0.33) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL24528652 0.95 KDM4E (0.32) KDM4EALDH1A1LMNA
SCHEMBL24528695 0.93 KDM4E (0.34) KDM4EALDH1A1LMNAMAPK1THRB
SCHEMBL24528677 0.93 KDM4E (0.34) KDM4EALDH1A1LMNAMAPK1TLR9
SCHEMBL24528715 0.90 KDM4E (0.38) KDM4EALDH1A1LMNAATMKMT2A
SCHEMBL29680698 0.90 KDM4E (0.38) KDM4EALDH1A1LMNAATMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed